BIOORGANIC CHEMISTRY (PRINT)
-
- Visão geral
-
- Metrics
-
- Identidade
-
- Ver todos
-
Visão geral
Qualis
código do país
tipo
publicação venue de
-
1,2,3-Triazolo[4,5-b]aminoquinolines: Design, synthesis, structure, acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) inhibitory activity, and molecular docking of novel modified tacrines.
139:106704.
2023-01-01
-
Design, synthesis and biological evaluation of antiparasitic dinitroaniline-ether phospholipid hybrids.
138:106615.
2023-01-01
-
New amides derived from sclareolide as anticholinesterase agents.
130:106249-12.
2023-01-01
-
C-phycocyanin decreases proliferation and migration of melanoma cells: In silico and in vitro evidences.
122:1.
2022-01-01
-
Caffeine improves the cytotoxic effect of dacarbazine on B16F10 murine melanoma cells.
120:105576.
2022-01-01
-
Chalcones from Angelica keiskei (ashitaba) inhibit key Zika virus replication proteins.
120:105649.
2022-01-01
-
Cholinesterase inhibitors assessment of aporphine alkaloids from Annona crassiflora and molecular docking studies.
1:105593-1.
2022-01-01
-
Click ferrocenyl-erlotinib conjugates active against erlotinib-resistant non-small cell lung cancer cells in vitro.
119:105514.
2022-01-01
-
Design, Synthesis and in vivo Evaluation of 1,4-dioxo-2-butenyl Aryl Amine Derivatives as a Promising Anti-inflammatory Drug Prototype.
1:105754.
2022-01-01
-
Discovery of (E)-4-styrylphenoxy-propanamide: A dual PPARα/γ partial agonist that regulates high-density lipoprotein-cholesterol levels, modulates adipogenesis, and improves glucose tolerance in diet-induced obese mice.
00:105600.
2022-01-01
-
Energy metabolism as a target for cyclobenzaprine: A drug candidate against Visceral Leishmaniasis.
1:106009-1.
2022-01-01
-
Iron chelation and inhibition of metallopeptidases mediate anti-Trichomonas vaginalis activity by a novel 8-hydroxyquinoline derivative.
125:105912.
2022-01-01
-
Novel Azine Linked Hybrids of 2-indolinone and Thiazolodinone Scaffolds as CDK2 inhibitors with potential anticancer activity: In Silico Design, Synthesis, Biological, Molecular Dynamics and Binding Free Energy Studies.
126:105884.
2022-01-01
-
Peptide inhibitors of angiotensin-I converting enzyme based on angiotensin (1-7) with selectivity for the C-terminal domain.
129:106204-227.
2022-01-01
-
Structural and biosynthetic studies of botrycinereic acid, a new cryptic metabolite from the fungus Botrytis cinerea.
127:105979.
2022-01-01
-
Synthesis of novel thiazolidinic-phthalimide derivatives evaluated as new multi-target antiepileptic agents.
119:105548-14.
2022-01-01
-
Unsaturated lipids modulating the interaction of the antileishmanial isolinderanolide E with models of cellular membranes.
124:105814.
2022-01-01
-
Violacein switches off low molecular weight tyrosine phosphatase and rewires mitochondria in colorectal cancer cells.
00:106000.
2022-01-01
-
4-chlorophenylthioacetone-derived thiosemicarbazones as potent antitrypanosomal drug candidates: investigations on the mode of action.
.:105018-..
2021-01-01
-
7-Amine-spiro[chromeno[4,3-b]quinoline-6,1?-cycloalkanes]: Synthesis and Cholinesterase Inhibitory Activity of Structurally Modified Tacrines.
108:104649.
2021-01-01
-
Accelerating the identification of subtype selective inhibitors via Three-Dimensional Biologically Relevant Spectrum (BRS-3D): The monoamine oxidase subtypes as a case study.
106:104503.
2021-01-01
-
Anti-inflammatory, ulcerogenic and platelet activation evaluation of novel 1,4-diaryl-1,2,3-triazole neolignan-celecoxib hybrids.
119:1-19.
2021-01-01
-
Antiamoebic effects of sesquiterpene lactones isolated from the zoanthid Palythoa aff. clavata.
108:104682.
2021-01-01
-
Antibacterial activity of a new monocarbonyl analog of curcumin MAC 4 is associated with divisome disruption.
1:104668-104672.
2021-01-01
-
Antioxidant and anti-sickling activity of glucal-based triazoles compounds - an in vitro and in silico study.
109:104709.
2021-01-01
-
Cathepsin K inhibitors based on 2-amino-1,3,4-oxadiazole derivatives.
.:104662-..
2021-01-01
-
Chalcones and their B-aryl analogues as myeloperoxidase inhibitors: In silico, in vitro and ex vivo investigations.
110:104773-104778.
2021-01-01
-
Design, synthesis and antibacterial activity of chalcones against MSSA and MRSA planktonic cells and biofilms.
116:105279.
2021-01-01
-
Discovery of 1,3,4,5-tetrasubstituted pyrazoles as anti-trypanosomatid agents: Identification of alterations in flagellar structure of L. amazonensis.
114:105082.
2021-01-01
-
Flavonoids from Pterogyne nitens as Zika virus NS2B-NS3 protease inhibitors.
109:104719.
2021-01-01
-
Hybrids of 4-Hydroxy Derivatives of Goniothalamin and Piplartine Bearing a Diester or a 1,2,3-Triazole Linker as Antiproliferative Agents.
116:105292-105292.
2021-01-01
-
Mefloquine synergism with anti-tuberculosis drugs and correlation to membrane effects: Biologic, spectroscopic and molecular dynamics simulations studies.
-:104786-104796.
2021-01-01
-
Natural-product-inspired design and synthesis of two series of compounds active against Trypanosoma cruzi: Insights into structure-activity relationship, toxicity, and mechanism of action.
118:105492-xx.
2021-01-01
-
New 5-carba-pterocarpans: Synthesis and preliminary antiproliferative activity on a panel of human cancer cells.
107:104584-104584.
2021-01-01
-
Novel inhibitors of the main protease enzyme of SARS-CoV-2 identified via molecular dynamics simulation-guided in vitro assay.
104862:104862.
2021-01-01
-
Quinazolinone dimers as a potential new class of safer Kv1 inhibitors: Overcoming hERG, Sodium and Calcium channel affinities.
115:105264.
2021-01-01
-
Scope and limitations of biocatalytic carbonyl reduction with white-rot fungi.
108:104651.
2021-01-01
-
Synthesis and In Vitro and In Silico Studies of 1H- and 2H-1,2,3-Triazoles as Antichagasic Agents.
00:105250.
2021-01-01
-
Synthesis and pharmacological evaluation of pomalidomide derivatives useful for sickle cell disease treatment.
114:105077.
2021-01-01
-
Synthesis of 3-aryl-4-(N-aryl)aminocoumarins via photoredox arylation and the evaluation of their biological activity.
114:105141.
2021-01-01
-
Synthesis of a novel glibenclamide-pioglitazone hybrid compound and its effects on glucose homeostasis in normal and insulin-resistant rats.
-:105157.
2021-01-01
-
Synthesis of chalcones derived from 1-naphthylacetophenone and evaluation of their cytotoxic and apoptotic effects in acute leukemia cell lines.
110:105315-105315.
2021-01-01
-
Synthesis of new α-Aryl-α-tetralones and α-Fluoro-α-aryl-α-tetralones, preliminary antiproliferative evaluation on drug resistant cell lines and in silico prediction of ADMETox properties.
110:104790.
2021-01-01
-
Synthesis, biological evaluation and molecular docking studies of novel 1,2,3-triazole-quinazolines as antiproliferative agents displaying ERK inhibitory activity.
113:104982.
2021-01-01
-
Targeting GRP receptor: design, synthesis and preliminary biological characterization of new non-peptide antagonists of bombesin.
109:104739.
2021-01-01
-
The role of remote flavin adenine dinucleotide pieces in the oxidative decarboxylation catalyzed by salicylate hydroxylase.
119:105561-X.
2021-01-01
-
oDissection of phospholipases A2 reveals multifaceted peptides targeting cancer cells, Leishmania and bacteria.
1:105041.
2021-01-01
-
Anti-Trypanosoma cruzi activity of costic acid isolated from Nectandra barbellata (Lauraceae) is associated with alterations in plasma membrane electric and mitochondrial membrane potentials..
95:103510-103538.
2020-01-01
-
Anti-cancer potential of sophoridine and its derivatives: Recent progress and future perspectives.
99:103863.
2020-01-01
-
Antileishmanial activity of 4-phenyl-1-[2-(phthalimido-2-yl)ethyl]-1H-1,2,3-triazole (PT4) derivative on Leishmania amazonensis and Leishmania braziliensis: In silico ADMET, in vitro activity, docking and molecular dynamic simulations.
105:104437.
2020-01-01
-
Antioxidant compounds from Banisteriopsis argyrophylla leaves as α-amylase, α-glucosidase, lipase, and glycation inhibitors.
105:104335.
2020-01-01
-
Batzelladine D and Norbatzelladine L Purified from Marine Sponge Monanchora arbuscula Induce the Reversal of Fluconazole.
105:104402-xxx.
2020-01-01
-
Calix[6]arene diminishes receptor tyrosine kinase lifespan in pancreatic cancer cells and inhibits their migration and invasion efficiency.
100:103881.
2020-01-01
-
Coumaric acid derivatives as tyrosinase inhibitors: Efficacy studies through in silico, in vitro and ex vivo approaches.
103:104108.
2020-01-01
-
Diaryl disulfides and thiosulfonates as combretastatin A-4 analogues: Synthesis, cytotoxicity and antitubulin activity.
101:104017.
2020-01-01
-
Differential lethal action of C17:2 and C17:0 anacardic acid derivatives in Trypanosoma cruzi - A mechanistic study.
102:104068-104073.
2020-01-01
-
Drug repurposing for the treatment of COVID-19: Pharmacological aspects and synthetic approaches.
106:104488-xxxx.
2020-01-01
-
Exploring the interaction between citrus flavonoids and phytopathogenic fungi through enzymatic activities.
1:104126-159.
2020-01-01
-
Geissoschizoline, a promising alkaloid for Alzheimer?s disease: Inhibition of human cholinesterases, anti-inflammatory effects and molecular docking.
.:104215.
2020-01-01
-
Interaction of dicentrinone, an antitrypanosomal aporphine alkaloid isolated from Ocotea puberula (Lauraceae), in cell membrane models at the air-water interface.
1:103978-1.
2020-01-01
-
Merulinic acid C overcomes gentamicin resistance in Enterococcus faecium.
000:103921.
2020-01-01
-
Modified pyrazole platinum(II) complex can circumvent albumin and glutathione: Synthesis, structure and cytotoxic activity.
00:103936.
2020-01-01
-
Molecular mechanism of action of new 1,4-naphthoquinones tethered to 1,2,3-1H-triazoles with cytotoxic and selective effect against oral squamous cell carcinoma.
.:103984.
2020-01-01
-
New antifungal ent-labdane diterpenes against Candida glabrata produced by microbial transformation of ent-polyalthic acid.
95:103560-103560.
2020-01-01
-
Novel pyranopyrazole derivatives comprising a benzoxazole core as antimicrobial inhibitors: Design, synthesis, microbial resistance and machine aided results.
100:103908.
2020-01-01
-
Optimization strategy of single-digit nanomolar cross-class inhibitors of mammalian and protozoa cysteine proteases.
101:104039.
2020-01-01
-
P2X7 receptor inhibition by 2-amino-3-aryl-1,4-naphthoquinones.
104:104278-104289.
2020-01-01
-
Pyrrole-2,5-dione Analogs as a Promising Antioxidant Agents: Microwave-assisted Synthesis, Bio-evaluation, SAR Analysis and DFT Studies / Interpretation.
106:104465.
2020-01-01
-
Stephalagine, an aporphine alkaloid from Annona crassiflora fruit peel, induces antinociceptive effects by TRPA1 and TRPV1 channels modulation in mice.
96:103562-..
2020-01-01
-
Synthesis and biological evaluation of 2?-Aminochalcone: a multi-target approach to find drug candidates to treat Alzheimer?s disease.
103:104201.
2020-01-01
-
Synthesis and evaluation of resveratrol derivatives as fetal hemoglobin inducers.
100:103948-103948.
2020-01-01
-
The antidiabetic drug lobeglitazone has the potential to inhibit PTP1B activity.
100:1.
2020-01-01
-
The insertion of functional groups in organic selenium compounds promote changes in mitochondrial parameters and raise the antibacterial activity.
98:103727-xx.
2020-01-01
-
Tolnaftate inhibits ergosterol production and impacts cell viability of Leishmania sp..
102:104056-104063.
2020-01-01
tem uma área de assunto
publisher
is open access
-
False
invalid format
is in DOAJ
-
False
invalid format
Metrics
2 year mean citedness
H index
i10 index
Identidade
ISSN-L
openalex identifier
-
https://openalex.org/S165482960
International Standard Serial Number (ISSN)